Puas yog Atorvastatin tuaj yeem yaj hauv dej?
Puas yog Atorvastatin tuaj yeem yaj hauv dej?

Video: Puas yog Atorvastatin tuaj yeem yaj hauv dej?

Video: Puas yog Atorvastatin tuaj yeem yaj hauv dej?
Video: pua yog tim tub aib pog ntawv by paj vuam thoj sonie thoj zoo siab yaj nkauj tawm tshiab 2022 2024, Lub Xya hli ntuj
Anonim

Chav kawm tshuaj: Tus neeg txo qis lipid, Statin

Ib yam nkaus, tib neeg nug, puas yog atorvastatin yaj hauv dej?

Atorvastatin calcium tsawg heev soluble nyob rau hauv distilled dej , pH 7.4 phosphate buffer, thiab acetonitrile, me ntsis soluble hauv ethanol thiab dawb soluble hauv methanol. LIPITOR ntsiav tshuaj muaj tshuaj atorvastatin calcium sib npaug rau 10, 20, 40 thiab 80 mg tshuaj atorvastatin.

Qhov thib ob, puas yog cov dej atorvastatin lossis cov rog yaj? Kev siv lipophilic, lossis rog - soluble statins xws li simvastatin thiab tshuaj atorvastatin tau cuam tshuam nrog txo qis kev pheej hmoo ntawm Parkinson's, thaum tsis muaj kev koom tes zoo li no rau hydrophilic, lossis dej - soluble , statins xws li pravastatin thiab rosuvastatin.

Xav txog qhov no, koj puas tuaj yeem yaj atorvastatin?

Nqa cov ntsiav tshuaj tag nrho. Ua tsis zuaj, tawg, zom, lossis yaj nws . Koj yuav noj cov tshuaj no nrog lossis tsis muaj zaub mov noj.

Yuav ua li cas koj thiaj li yaj simvastatin?

Simvastatin yog me ntsis soluble hauv dej tsis. Txog qhov siab tshaj plaws nyob hauv cov dej tsis zoo, simvastatin yuav tsum xub ua yaj hauv DMSO thiab tom qab ntawd diluted nrog cov dej tsis tuaj yeem xaiv. Simvastatin muaj qhov sib tov kwv yees li 0.5 mg/ml hauv 1: 1 daws ntawm DMSO: PBS (pH 7.2) siv txoj hauv kev no.

Pom zoo: