Dab tsi tshwm sim thaum benzodiazepines khi rau lawv cov receptors hauv lub hlwb?
Dab tsi tshwm sim thaum benzodiazepines khi rau lawv cov receptors hauv lub hlwb?

Video: Dab tsi tshwm sim thaum benzodiazepines khi rau lawv cov receptors hauv lub hlwb?

Video: Dab tsi tshwm sim thaum benzodiazepines khi rau lawv cov receptors hauv lub hlwb?
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Benzodiazepines khi mus rau stereospecific benzodiazepine receptors ntawm lub hauv paus paj hlwb (CNS) GABA A cov receptors , ua rau muaj zog neuronal membrane permeability rau chloride ions. GABA A tus txais agonism los ntawm benzodiazepines ua rau sedative, hypnotic, anxiolytic, antiepileptic, thiab cov leeg so kom txaus.

Kuj paub yog, dab tsi yog ib feem ntawm lub hlwb puas benzodiazepines cuam tshuam?

Cov tshuaj benzodiazepines nyuaj siab rau hauv nruab nrab lub paj hlwb (CNS). Cov CNS kev nyuaj siab no cuam tshuam cov lub hlwb neurotransmitter GABA (gamma-aminobutyric acid). GABA qis lub hlwb kev ua, uas ua rau koj tsaug zog lossis nyob ntsiag to.

Tsis tas li ntawd, cov receptors twg hauv lub hlwb ua sedative hypnotic agents khi rau? Sedative - Hypnotics Zoo tag nrho cov tshuaj sedative , hypnotic thiab anxiolytic cov neeg sawv cev khi rau GABA moieties ntawm benzodiazepine tus txais.

Kuj paub, dab tsi yog lub tswv yim ntawm kev ua ntawm benzodiazepines?

Cov tshuaj benzodiazepines txhim kho cov nyhuv ntawm cov neurotransmitter gamma-aminobutyric acid (GABA) ntawm GABAA receptor, ua rau muaj sedative, hypnotic (tsaug zog inducing), anxiolytic (anti-ntxhov siab vim), anticonvulsant, thiab cov leeg so kom txaus zog.

Puas Benzos cuam tshuam rau dopamine?

Txawm li cas los xij, tsis zoo li cov tshuaj stimulant, benzodiazepines tsis txhob nce dopamine qib ncaj qha. Hloov chaw, lawv txo qis cov txiaj ntsig ib txwm muaj ntawm lwm cov neurotransmitter hu ua GABA (gamma-aminobutyric acid), uas feem ntau pab ua kom qeeb ntawm cov paj hlwb (neurons) uas tsim tawm. dopamine.

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