Dab tsi yog ntshiab opioid agonists?
Dab tsi yog ntshiab opioid agonists?

Video: Dab tsi yog ntshiab opioid agonists?

Video: Dab tsi yog ntshiab opioid agonists?
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Ntshiab opioid agonists (piv txwv li, morphine, hydromor-phone, fentanyl) txhawb nqa µ receptors thiab yog cov tshuaj muaj zog tshaj plaws.

Ntawm no, dab tsi yog ib qho opioid agonist?

Piv txwv ntawm tag nrho agonists suav nrog codeine, fentanyl, heroin, hydrocodone, methadone, morphine, thiab oxycodone. Thiab, qee qhov cov tshuaj opioids yog agonists ntawm 1 lossis ntau dua opioid receptors tab sis kuj yog antagonists ntawm lwm tus opioid receptors . Cov ntsiab lus ntawm cov teebmeem receptor rau agonists /antagonists tuaj yeem pom hauv Table 4.

Ib yam nkaus, cov tshuaj twg yog agonist thiab antagonist? Piv txwv ntawm tag nrho agonists yog heroin, oxycodone, methadone, hydrocodone, morphine, opium thiab lwm yam. Ib tus yeeb ncuab yog a tshuaj uas thaiv opioids los ntawm kev txuas mus rau cov neeg txais tshuaj opioid yam tsis tau qhib lawv. Antagonists ua rau tsis muaj cov nyhuv opioid thiab thaiv tag nrho agonist cov tshuaj opioids. Piv txwv yog naltrexone thiab naloxone.

Ib sab saum toj no, dab tsi yog cov antagonists rau cov tshuaj opioid?

Ob qhov feem ntau siv hauv nruab nrab ua yeeb yam opioid receptor antagonists yog naloxone thiab naltrexone . Naloxone los rau hauv cov hlab ntshav, intramuscular thiab intranasal formulations, thiab tau pom zoo los ntawm FDA rau kev siv tshuaj opioid ntau dhau, thiab kev thim rov qab ntawm kev nyuaj siab ua pa cuam tshuam nrog kev siv opioid.

Puas yog hydrocodone tag nrho agonist?

Ib agonist yog ib yam tshuaj uas ua kom muaj qee tus neeg txais hauv lub hlwb. Tag nrho agonist opioids qhib lub opioid receptors hauv lub hlwb tag nrho ua rau puv cov nyhuv opioid. Piv txwv ntawm tag nrho agonists yog heroin, oxycodone, tshuaj txiav yeeb, hydrocodone , morphine, opium thiab lwm yam.

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