Alpha 2 agonist ua dab tsi?
Alpha 2 agonist ua dab tsi?

Video: Alpha 2 agonist ua dab tsi?

Video: Alpha 2 agonist ua dab tsi?
Video: Autonomic Pharmacology (Ar) - Lec 02 - Adrenergic Receptors 2024, Lub Xya hli ntuj
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α2 agonist : txwv tsis pub ua haujlwm adenylyl cyclase, txo qis kev ua haujlwm ntawm vasomotor nruab nrab-nruab nrab CNS ua kom; siv raws li antihypertensive, sedative & kev kho mob ntawm kev quav yeeb quav tshuaj thiab cov tsos mob tshem tawm cawv).

Tsis tas li ntawd, alpha 2 agonists cuam tshuam li cas rau ntshav siab?

Alpha 2 receptors nyob rau hauv lub paj hlwb thiab nyob ib puag ncig cuam tshuam kev ua siab zoo thiab yog li qis ntshav siab . Alpha 2 tus txais agonists xws li clonidine lossis guanabenz txo qis hauv nruab nrab thiab cov khoom nruab nrog sab hauv uas muaj kev nkag siab zoo thiab ntawm cov khoom siv ib puag ncig presynaptic cov neeg txais yuav txo qis kev tso tawm cov hlab ntsha ib leeg.

Tom qab ntawd, lo lus nug yog, Alpha 2 ua rau vasoconstriction? Lub luag haujlwm ntawm alpha ( 2 ) -AR tsev neeg tau paub ntev los suav nrog presynaptic inhibition ntawm kev tso tawm cov tshuaj xa mus rau lub cev, txo qis kev nkag siab zoo ntawm cov tsheb khiav mus los, vasodilation thiab vasoconstriction . Cov lus teb nyuaj no tau kho kom haum xeeb los ntawm ib ntawm peb hom subtypes uas txhua qhov tshwj xeeb cuam tshuam rau ntshav siab thiab ntshav ntws.

Tsis tas li, tshuaj alpha 2 agonist yog dab tsi?

Alpha - 2 agonists . Clonidine (Catapres®) Clonidine thaj (Catapres -TTS®) Methyldopa (Aldomet®) Tizanidine (Zanaflex®) - siv los ua leeg nqaij.

Tus alpha agonist ua haujlwm li cas?

Alpha -adrenoceptor tus neeg mob agonists ( α - agonists ) khi rau α -receptors ntawm cov leeg leeg leeg thiab ua kom sib zog ua kom sib zog thiab ua kom lub vasoconstriction, yog li ua raws li qhov cuam tshuam ntawm kev nkag siab zoo adrenergic ua kom cov hlab ntsha mus rau cov hlab ntsha.

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